A General Method for Suzuki–Miyaura Coupling Reactions Using Lithium Triisopropyl Borates

Conditions for the Suzuki–Miyaura coupling of lithium triisopropyl borates are reported, as well as a procedure for a one-pot lithiation, borylation, and subsequent Suzuki–Miyaura coupling of various heterocycles with aryl halides. These borate species are much more stable toward protodeboronation t...

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Bibliographic Details
Main Authors: Buchwald, Stephen Leffler, Oberli, Matthias
Other Authors: David H. Koch Institute for Integrative Cancer Research at MIT
Format: Article
Published: American Chemical Society (ACS) 2013
Online Access:http://hdl.handle.net/1721.1/81947

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